SCHEMBL7344698

SCHEMBL7344698

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(N(C)C)CC2)ccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
KDM4E B2RXH2 7/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
TMPRSS2 O15393 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344697 0.91 ALDH1A1 (0.39) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL7335732 0.90 ALDH1A1 (0.43) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL7343093 0.88 POLB (0.39) ALDH1A1KDM4ELMNAMAPTTP53
SCHEMBL7780726 0.88 POLB (0.38) KDM4ELMNAPOLBTHRATHRB
SCHEMBL7345680 0.85 ALDH1A1 (0.43) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL7781259 0.84 NPC1 (0.42) KDM4EKMT2AMEN1POLBRAB9A
SCHEMBL7339114 0.83 AVPR2 (0.42) ALDH1A1LMNAMAPTPOLBRAB9A
SCHEMBL7373593 0.83 ALDH1A1 (0.43) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL7334833 0.82 ALDH1A1 (0.43) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL7379368 0.82 AVPR2 (0.51) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed
EP-0832061-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-01 EP disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed