SCHEMBL7344733

SCHEMBL7344733

CC(C)(C)OC(=O)NC(Cc1cccs1)C(=O)CSCc1ccco1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.54
CTSS P25774 3/20 0.54
ALDH1A1 P00352 7/20 0.50
HPGD P15428 4/20 0.50
HSD17B10 Q99714 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
MAPT P10636 2/20 0.50
PPARG P37231 5/20 0.41
PPARA Q07869 5/20 0.41
PPARD Q03181 2/20 0.40
CTSL P07711 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ACE P12821 1/20 0.38
ADAM17 P78536 1/20 0.38
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344725 1.00 CTSK (0.54) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7340544 0.85 ACE (0.54) CTSKCTSSPPARGPPARAPPARD
SCHEMBL7340534 0.85 ACE (0.54) CTSKCTSSPPARGPPARAPPARD
SCHEMBL7349733 0.84 CTSK (0.50) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7349722 0.84 CTSK (0.50) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7340555 0.83 CTSK (0.51) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7340560 0.83 CTSK (0.51) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7349130 0.83 PPARG (0.52) CTSKCTSSALDH1A1HPGDHSD17B10
SCHEMBL7345612 0.83 CTSS (0.51) CTSKCTSSALDH1A1HPGDPPARG
SCHEMBL7345598 0.83 CTSS (0.51) CTSKCTSSALDH1A1HPGDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603873-B1 Aminoketone derivatives MITSUBISHI CHEM CORP (JP) 1998-04-15 EP disclosed
US-5424325-A Inibitors of thiol protease and may be used as therapeutic agents for treating muscular dystrophy, cataracts, strokes MITSUBISHI KASEI CORPORATION (JP) 1995-06-13 US disclosed
EP-0603873-A1 Aminoketone derivatives Mitsubishi Chemical Corporation (JP) 1994-06-29 EP disclosed