SCHEMBL7344748

SCHEMBL7344748

CNS(=O)(=O)NCCNC(=O)[C@@H](C[C@H](O)[C@H](C)NC(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.38
CA2 P00918 4/20 0.37
CTSS P25774 4/20 0.36
CTSK P43235 4/20 0.36
CAPN1 P07384 1/20 0.36
CA1 P00915 1/20 0.35
CA7 P43166 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
REN P00797 3/20 0.32
CTSD P07339 1/20 0.32
CTSE P14091 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259871 0.83 CYP2D6 (0.40) CYP2D6CA2CTSSCTSKCAPN1
SCHEMBL9263938 0.82 CYP2D6 (0.42) CYP2D6CA2CTSSCTSKCAPN1
SCHEMBL7412829 0.77 CYP2D6 (0.42) CYP2D6CA2CTSSCTSKCAPN1
SCHEMBL9262937 0.76 CYP2D6 (0.41) CYP2D6CA2CTSSCTSKCA1
SCHEMBL9270675 0.75 CTSL (0.40) CYP2D6CTSSCTSKCAPN1CTSL
SCHEMBL9287940 0.74 CD274 (0.47) CTSKREN
SCHEMBL7345146 0.73 CYP2D6 (0.48) CYP2D6CA2CTSSCTSKCA1
SCHEMBL9286028 0.72 ALDH1A1 (0.47) REN
SCHEMBL7410615 0.72 KMT2A (0.51) CA2RENCTSDCTSE
SCHEMBL7417716 0.71 BACE1 (0.52) RENCTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389647-A A prodrugs as hypotensive agents, treating congestive heart failure, urogenital disorders, vision defects ABBOTT LABORATORIES (US) 1995-02-14 US disclosed
US-5244910-A Treating hypertension, congestive heart failure ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
WO-1992003429-A1 RENIN INHIBITORS ABBOTT LABORATORIES (US) 1992-03-05 WO disclosed