SCHEMBL9259871

SCHEMBL9259871

CNS(=O)(=O)NNC(=O)[C@@H](C[C@H](O)[C@H](C)NC(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.40
CA2 P00918 3/20 0.37
CA1 P00915 2/20 0.37
CA7 P43166 2/20 0.37
CTSK P43235 5/20 0.36
CTSS P25774 4/20 0.36
CTSL P07711 2/20 0.34
CTSB P07858 1/20 0.34
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
CA12 O43570 1/20 0.33
CA14 Q9ULX7 1/20 0.33
REN P00797 1/20 0.31
CTSD P07339 1/20 0.31
CTSE P14091 1/20 0.31
CAPN1 P07384 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9262937 0.88 CYP2D6 (0.41) CYP2D6CA2CA1CA7CTSK
SCHEMBL7344748 0.83 CYP2D6 (0.38) CYP2D6CA2CA1CA7CTSK
SCHEMBL7345146 0.76 CYP2D6 (0.48) CYP2D6CA2CA1CA7CTSK
SCHEMBL9263938 0.75 CYP2D6 (0.42) CYP2D6CA2CA1CA7CTSK
SCHEMBL7412829 0.75 CYP2D6 (0.42) CYP2D6CA2CA1CA7CTSK
SCHEMBL19790304 0.72 CA1 (0.53) CYP2D6CA2CA1CA7CTSK
SCHEMBL14923535 0.72 CA1 (0.53) CYP2D6CA2CA1CA7CTSK
SCHEMBL9270675 0.69 CTSL (0.40) CYP2D6CTSKCTSSCTSLCTSB
SCHEMBL7417716 0.69 BACE1 (0.52) RENCTSDCTSE
SCHEMBL7419674 0.68 REN (0.45) CYP2D6CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389647-A A prodrugs as hypotensive agents, treating congestive heart failure, urogenital disorders, vision defects ABBOTT LABORATORIES (US) 1995-02-14 US disclosed
US-5244910-A Treating hypertension, congestive heart failure ABBOTT LABORATORIES (US) 1993-09-14 US disclosed