SCHEMBL7344814

SCHEMBL7344814

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2C(=O)c3ccccc3C2=O)C1c1c(Cl)cccc1[N+](=O)[O-]

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.57
CYP1A2 P05177 6/20 0.50
CYP2C9 P11712 6/20 0.50
HIF1A Q16665 6/20 0.50
KMT2A Q03164 6/20 0.50
CYP3A4 P08684 5/20 0.50
CYP2C19 P33261 5/20 0.50
MAPT P10636 5/20 0.50
ADORA3 P0DMS8 4/20 0.50
LMNA P02545 4/20 0.50
ABCB11 O95342 3/20 0.50
SCN1A P35498 3/20 0.50
SCN5A Q14524 3/20 0.50
SCN2A Q99250 3/20 0.50
SCN3A Q9NY46 3/20 0.50
KDM4E B2RXH2 3/20 0.50
CYP2D6 P10635 3/20 0.50
TSHR P16473 3/20 0.50
NFKB1 P19838 3/20 0.50
THPO P40225 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346372 0.94 HSD17B10 (0.62) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7347242 0.87 ADORA3 (0.69) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7350118 0.86 HSD17B10 (0.61) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7343960 0.85 ADORA3 (0.50) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7350016 0.84 HSD17B10 (0.56) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7348263 0.83 HSD17B10 (0.66) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL7347116 0.82 HSD17B10 (0.56) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL9673018 0.82 CYP2C9 (0.68) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL9674378 0.82 ADORA3 (0.66) HSD17B10CYP1A2CYP2C9HIF1AKMT2A
SCHEMBL10918103 0.81 MAPT (0.70) CYP1A2CYP2C9HIF1AKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed