SCHEMBL7346372

SCHEMBL7346372

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2C(=O)c3ccccc3C2=O)C1c1c([N+](=O)[O-])cccc1[N+](=O)[O-]

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.62
MAPT P10636 6/20 0.54
ADORA3 P0DMS8 5/20 0.54
CYP1A2 P05177 5/20 0.54
KMT2A Q03164 5/20 0.54
HIF1A Q16665 4/20 0.54
CYP3A4 P08684 4/20 0.54
CYP2C9 P11712 4/20 0.54
CYP2C19 P33261 4/20 0.54
TDP1 Q9NUW8 4/20 0.54
LMNA P02545 3/20 0.54
OPRM1 P35372 3/20 0.54
CYP2D6 P10635 3/20 0.54
ABCC4 O15439 2/20 0.54
CACNA1F O60840 2/20 0.54
ABCB11 O95342 2/20 0.54
ADORA2A P29274 2/20 0.54
ADORA1 P30542 2/20 0.54
SCN1A P35498 2/20 0.54
HTR2B P41595 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344814 0.94 HSD17B10 (0.57) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL7347242 0.91 ADORA3 (0.69) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL9674378 0.85 ADORA3 (0.66) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL9672675 0.85 ADORA3 (0.65) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL7350843 0.85 MAPT (0.70) MAPTADORA3CYP1A2KMT2AHIF1A
SCHEMBL10918103 0.85 MAPT (0.70) MAPTADORA3CYP1A2KMT2AHIF1A
SCHEMBL7350016 0.84 HSD17B10 (0.56) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL9674762 0.84 ADORA3 (0.64) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL7346357 0.83 CYP1A2 (0.54) HSD17B10MAPTADORA3CYP1A2KMT2A
SCHEMBL7341132 0.83 HSD17B10 (0.59) HSD17B10MAPTADORA3CYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed