SCHEMBL7345235

SCHEMBL7345235

COc1ccc2cc(C3(C)C=CC=CN3)ccc2n1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.34
LMNA P02545 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CDK6 Q00534 1/20 0.31
NCF1 P14598 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270869 0.67 NCF1 (0.41) ADORA1HDAC3HDAC4HDAC1HDAC2
SCHEMBL423324 0.65 CYP1A2 (0.59) NCF1
SCHEMBL30081479 0.64 BACE1 (0.53) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL727654 0.64 BACE1 (0.53) ADORA1HDAC3HDAC4HDAC1HDAC2
SCHEMBL19330216 0.64 HTR3A (0.45) ADORA1HDAC3HDAC4HDAC1HDAC2
SCHEMBL29768705 0.64 ESR1 (0.50) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL7270843 0.64 APP (0.41) ADORA1HDAC3HDAC4HDAC1HDAC2
SCHEMBL1238150 0.64 ESR1 (0.50) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL21698711 0.64 KDM4E (0.58) LMNAHDAC3HDAC4HDAC1HDAC2
SCHEMBL16751340 0.63 PDE10A (0.46) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5141931-A 5-Quinolinylpyridinones, cardiotonic compositions and methods STERLING WINTHROP INC. (US) 1992-08-25 US disclosed