SCHEMBL7345238

SCHEMBL7345238

COc1ccc2cc(-c3cccnc3C)ccc2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.52
PDE2A O00408 3/20 0.52
ADORA1 P30542 1/20 0.44
BACE1 P56817 2/20 0.43
CTSD P07339 1/20 0.43
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
ABL1 P00519 2/20 0.42
TGFBR1 P36897 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
DHODH Q02127 1/20 0.40
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
MAT2A P31153 1/20 0.38
JAK3 P52333 2/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15730144 0.82 POLB (0.47) BACE1CTSDNPC1POLBRAB9A
SCHEMBL15730171 0.81 NPC1 (0.67) NPC1POLBRAB9AABL1TGFBR1
SCHEMBL15730178 0.80 CYP11B2 (0.56) NPC1RAB9AABL1
SCHEMBL15730261 0.76 CYP2A6 (0.54) PDE10APDE2AMKNK1MKNK2JAK2
SCHEMBL16805031 0.76 ABL1 (0.52) ADORA1NPC1POLBRAB9AABL1
SCHEMBL7264558 0.74 CYP11B2 (0.64) PDE10APDE2AABL1MKNK1MKNK2
SCHEMBL16573997 0.74 PDGFRB (0.46) PDE10APDE2AADORA1BACE1NPC1
SCHEMBL12695592 0.74 BACE1 (0.57) ADORA1BACE1NPC1RAB9APDGFRB
SCHEMBL15730608 0.74 ALDH1A1 (0.58) NPC1POLBRAB9AABL1TGFBR1
SCHEMBL7270915 0.73 ADORA1 (0.42) PDE10APDE2AADORA1NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5141931-A 5-Quinolinylpyridinones, cardiotonic compositions and methods STERLING WINTHROP INC. (US) 1992-08-25 US disclosed