SCHEMBL7345562

SCHEMBL7345562

COc1ccc(OC[C]=O)c(OC)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA7 P43166 1/20 0.59
CA9 Q16790 1/20 0.59
CA14 Q9ULX7 1/20 0.59
ALDH1A1 P00352 6/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADRA1A P35348 2/20 0.44
ADRA2A P08913 1/20 0.44
HSD17B10 Q99714 1/20 0.44
APLNR P35414 1/20 0.43
CYP1A1 P04798 4/20 0.43
CYP1A2 P05177 4/20 0.43
CYP1B1 Q16678 4/20 0.43
MAPT P10636 2/20 0.43
CYP3A4 P08684 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641220 0.87 CA2 (0.55) CA12CA1CA2CA7CA9
SCHEMBL9130705 0.84 GAA (0.47) CA12CA1CA2CA7CA9
SCHEMBL20985765 0.82 CA12 (0.59) CA12CA1CA2CA7CA9
SCHEMBL2089706 0.79 CA12 (0.65) CA12CA1CA2CA7CA9
SCHEMBL9911561 0.79 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL8888440 0.77 CA12 (0.68) CA12CA1CA2CA7CA9
SCHEMBL514580 0.77 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL5255563 0.77 MAOA (0.49) ALDH1A1LMNAHTTSMN1; SMN2HSD17B10
SCHEMBL15094776 0.77 APLNR (0.46) CA12CA1CA2CA7CA9
SCHEMBL5134647 0.77 BCHE (0.39) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
EP-0450097-A1 BENZOHETEROCYCLIC COMPOUNDS. OTSUKA PHARMA CO LTD (JP) 1991-10-09 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed