SCHEMBL7345718

SCHEMBL7345718

O=C1CCCCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LMNA P02545 3/20 0.49
USP2 O75604 2/20 0.49
PDE4B Q07343 1/20 0.49
PDE4D Q08499 1/20 0.49
TP53 P04637 1/20 0.49
TSHR P16473 1/20 0.49
MAPT P10636 4/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
AVPR2 P30518 6/20 0.49
AVPR1A P37288 5/20 0.49
OXTR P30559 2/20 0.49
MEN1 O00255 2/20 0.49
POLB P06746 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 2/20 0.48
GAA P10253 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990464 0.96 ALDH1A1 (0.52) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL7352575 0.93 ALDH1A1 (0.56) ALDH1A1LMNAUSP2TP53TSHR
SCHEMBL7351070 0.86 AVPR2 (0.67) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL6959618 0.85 AVPR2 (0.68) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL7352245 0.84 MEN1 (0.50) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL6968459 0.84 BCHE (0.56) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL7352139 0.84 AVPR2 (0.52) ALDH1A1LMNAUSP2MAPTAVPR2
SCHEMBL6961949 0.82 MAPT (0.48) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL6961951 0.82 MAPT (0.48) ALDH1A1LMNAUSP2PDE4BPDE4D
SCHEMBL7347078 0.82 AVPR2 (0.71) ALDH1A1LMNAUSP2TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed