SCHEMBL7352575

SCHEMBL7352575

O=C1CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
LMNA P02545 3/20 0.56
USP2 O75604 1/20 0.56
TP53 P04637 1/20 0.56
TSHR P16473 1/20 0.56
HTT P42858 2/20 0.53
HPGD P15428 2/20 0.50
BCHE P06276 1/20 0.49
P2RX4 Q99571 1/20 0.49
MAPT P10636 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
STING1 Q86WV6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990464 0.94 ALDH1A1 (0.52) ALDH1A1LMNAUSP2TP53TSHR
SCHEMBL7345718 0.93 ALDH1A1 (0.49) ALDH1A1LMNAUSP2TP53TSHR
SCHEMBL8562104 0.86 HPGD (0.58) ALDH1A1LMNAUSP2HTTHPGD
SCHEMBL842907 0.83 HPGD (0.64) ALDH1A1LMNAUSP2TP53TSHR
SCHEMBL21160915 0.82 HPGD (0.49) ALDH1A1LMNAHPGDBCHEP2RX4
SCHEMBL3044124 0.82 KCNN4 (0.68) ALDH1A1HTTHPGDBCHEP2RX4
SCHEMBL7352245 0.81 MEN1 (0.50) ALDH1A1LMNAUSP2HTTHPGD
SCHEMBL7348630 0.81 L3MBTL1 (0.46) ALDH1A1HTTHPGDBCHEP2RX4
SCHEMBL7349991 0.81 L3MBTL1 (0.46) ALDH1A1LMNAUSP2TP53TSHR
SCHEMBL7351134 0.81 AVPR2 (0.59) ALDH1A1LMNAUSP2TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1048484-C A process for preparing a composition containing benzoheterocycles OTSUKA PHARMA CO LTD (JP) 2000-01-19 CN disclosed
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
CN-1107146-A A process for preparing a composition containing benzoheterocycles OTSUKA PHARMA CO LTD (JP) 1995-08-23 CN disclosed
CN-1027505-C Process for preparing benzoheterocyclic compounds OTSUKA PHARMA CO LTD (JP) 1995-01-25 CN disclosed
EP-0450097-A1 BENZOHETEROCYCLIC COMPOUNDS. OTSUKA PHARMA CO LTD (JP) 1991-10-09 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed
CN-1051038-A BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1991-05-01 CN disclosed