SCHEMBL7345842

SCHEMBL7345842

COc1c(C(=O)c2ccccc2OCCCN2C(=O)c3ccccc3C2=O)ccc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(N(C)C)CC2)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
LMNA P02545 5/20 0.35
MAPT P10636 3/20 0.35
HTT P42858 3/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ACHE P22303 1/20 0.33
AVPR2 P30518 1/20 0.33
AVPR1A P37288 1/20 0.33
AVPR1B P47901 1/20 0.33
HTR4 Q13639 2/20 0.33
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780715 0.94 ALDH1A1 (0.39) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL7778674 0.86 KMT2A (0.42) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL7340123 0.85 KMT2A (0.36) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL7339161 0.85 CDK1 (0.35) LMNAMAPTHTTCDK1CDK4
SCHEMBL7340129 0.85 KMT2A (0.36) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL7340721 0.83 AVPR2 (0.39) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL7345832 0.82 AVPR2 (0.46) ALDH1A1LMNAMEN1KMT2AAVPR2
SCHEMBL7337098 0.81 CDK1 (0.36) CDK1CDK4CCND1CDK2ACHE
SCHEMBL7340552 0.80 CDK1 (0.36) LMNAMAPTHTTCDK1CDK4
SCHEMBL7478475 0.79 CBX7 (0.38) ALDH1A1MAPTHPGDMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed