SCHEMBL7345932

SCHEMBL7345932

NC(=S)c1cc2c([nH]c1=O)CCc1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.40
TYMS P04818 3/20 0.39
SRD5A1 P18405 2/20 0.38
SRD5A2 P31213 1/20 0.38
NOTUM Q6P988 1/20 0.38
MIF P14174 1/20 0.36
PDPK1 O15530 1/20 0.35
PARP1 P09874 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP11 Q9NR21 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
RAB9A P51151 2/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347752 0.92 ALDH1A1 (0.42) CES1TYMSSRD5A1SRD5A2NOTUM
SCHEMBL7336750 0.89 CYP1A2 (0.36) CES1SRD5A2PARP1KDM4EALDH1A1
SCHEMBL7339006 0.87 NOTUM (0.44) CES1TYMSSRD5A1SRD5A2NOTUM
SCHEMBL7342355 0.86 CES1 (0.40) CES1TYMSSRD5A1SRD5A2NOTUM
Hydrochloric Acid SCHEMBL7337010 0.84 CES1 (0.39) CES1TYMSSRD5A1SRD5A2NOTUM
SCHEMBL7340881 0.82 KDM4E (0.54) CES1SRD5A1SRD5A2NOTUMKDM4E
SCHEMBL7338264 0.79 TYMS (0.46) CES1TYMSSRD5A1SRD5A2PDPK1
SCHEMBL7336897 0.79 CES1 (0.44) CES1TYMSSRD5A1SRD5A2MIF
SCHEMBL7345410 0.78 KDM4E (0.48) CES1TYMSSRD5A1SRD5A2L3MBTL1
SCHEMBL7345933 0.77 SRD5A1 (0.38) CES1TYMSSRD5A1SRD5A2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4511569-A Tricyclic lactams and derivatives useful in increasing cardiac contractility SCHERING CORPORATION (US) 1985-04-16 US disclosed
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed