SCHEMBL7345960

SCHEMBL7345960

O=C(CCN(Cc1ccccc1)Cc1ccccc1)c1ccc(Br)cc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
DGAT1 O75907 1/20 0.44
HDAC3 O15379 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
NCOR2 Q9Y618 2/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 1/20 0.43
PDPK1 O15530 1/20 0.41
KMT2A Q03164 2/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GPR27 Q9NS67 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PARP15 Q460N3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352468 0.84 HTT (0.44) TMEM97SIGMAR1HDAC3HDAC1HDAC2
SCHEMBL7351073 0.82 HDAC3 (0.44) TMEM97SIGMAR1HDAC3HDAC1HDAC2
SCHEMBL13083453 0.80 KDM4E (0.49) KMT2AMEN1MAPTL3MBTL1
SCHEMBL7347710 0.76 KMT2A (0.49) TMEM97SIGMAR1DGAT1HDAC3HDAC1
SCHEMBL7346997 0.76 MEN1 (0.42) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL3280774 0.75 TMEM97 (0.56) TMEM97SIGMAR1DGAT1HDAC3HDAC1
SCHEMBL691531 0.73 DGAT1 (0.61) TMEM97SIGMAR1DGAT1NPC1KMT2A
SCHEMBL29993519 0.73 DGAT1 (0.61) TMEM97SIGMAR1DGAT1NPC1KMT2A
SCHEMBL3054837 0.72 DGAT1 (0.56) TMEM97SIGMAR1DGAT1NPC1PDPK1
SCHEMBL11900526 0.72 DGAT1 (0.56) TMEM97SIGMAR1DGAT1HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0972764-A1 Aminoalcohols and aminoketones as CNS active agents Universita Degli Studi di Firenze (IT) 2000-01-19 EP claimed
EP-0972764-A1 Aminoalcohols and aminoketones as CNS active agents Universita Degli Studi di Firenze (IT) 2000-01-19 EP disclosed