SCHEMBL7346902

SCHEMBL7346902

CC(C)(CN)[C@@H](C(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KMT2A Q03164 2/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LTA4H P09960 1/20 0.43
LAP3 P28838 1/20 0.43
SLC15A1 P46059 1/20 0.42
SLC1A3 P43003 2/20 0.42
SLC1A2 P43004 2/20 0.42
SLC1A1 P43005 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27691294 1.00 ALDH1A1 (0.49) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL7212486 0.86 ALDH1A1 (0.50) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL31294203 0.85 ALDH1A1 (0.56) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL6946125 0.85 ALDH1A1 (0.56) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL6946124 0.84 ALDH1A1 (0.62) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL6703901 0.82 ALDH1A1 (0.49) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL7208161 0.80 ALDH1A1 (0.53) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL14943541 0.78 ALDH1A1 (0.59) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL27780855 0.77 SYK (0.44) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL29008750 0.76 ALDH1A1 (0.53) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101133060-B Enzyme inhibitors CHROMA THERAPEUTICS LTD 2013-06-05 CN disclosed
CN-102161656-B Aspartic acid-specific caspase inhibitors and uses thereof VERTEX PHARMA 2013-02-20 CN disclosed
US-5338726-A Hypotensive agents, antiulcer agents ABBOTT LABORATORIES (US) 1994-08-16 US disclosed
EP-0569487-A4 1994-04-27 EP disclosed
EP-0569487-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS ABBOTT LABORATORIES (US) 1993-11-18 EP disclosed
WO-1992013545-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS ABBOTT LABORATORIES (US) 1992-08-20 WO disclosed