SCHEMBL7347334

SCHEMBL7347334

CC(N=C(NC#N)Nc1cccnc1)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.58
ABCC9 O60706 14/20 0.56
KCNJ11 Q14654 14/20 0.56
ABCC8 Q09428 8/20 0.56
KCNJ8 Q15842 8/20 0.56
CYP3A4 P08684 3/20 0.56
KMT2A Q03164 2/20 0.56
CYP1A2 P05177 2/20 0.56
MEN1 O00255 1/20 0.56
CYP2D6 P10635 1/20 0.56
NAMPT P43490 1/20 0.51
CYP2C9 P11712 1/20 0.48
ALOX15 P16050 1/20 0.48
NFKB1 P19838 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347346 0.87 ABCC9 (0.50) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL7352529 0.85 ABCC9 (0.48) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL7349440 0.85 ABCC9 (0.58) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL7348943 0.83 ABCC9 (0.54) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL9456841 0.81 ABCC9 (0.73) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7360174 0.81 NAMPT (0.50) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL8919354 0.80 ABCC9 (0.53) P2RX7ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL9297479 0.79 ABCC9 (0.71) P2RX7ABCC9KCNJ11CYP3A4CYP1A2
SCHEMBL9297483 0.79 ABCC9 (0.71) P2RX7ABCC9KCNJ11CYP3A4CYP1A2
SCHEMBL11157791 0.77 ABCC9 (0.70) P2RX7ABCC9KCNJ11ABCC8KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP claimed
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP disclosed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US disclosed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO disclosed