SCHEMBL7347346

SCHEMBL7347346

CC(N=C(NC#N)Nc1cccnc1)c1cccc(I)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 14/20 0.50
KCNJ11 Q14654 14/20 0.50
ABCC8 Q09428 8/20 0.50
KCNJ8 Q15842 8/20 0.50
CYP3A4 P08684 3/20 0.50
CYP1A2 P05177 2/20 0.50
MEN1 O00255 1/20 0.50
CYP2D6 P10635 1/20 0.50
KMT2A Q03164 1/20 0.50
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
ADRB3 P13945 1/20 0.50
P2RX7 Q99572 3/20 0.48
TBXA2R P21731 1/20 0.47
TBXAS1 P24557 1/20 0.47
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
NFKB1 P19838 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347334 0.87 P2RX7 (0.58) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7352529 0.85 ABCC9 (0.48) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7347341 0.79 ADRB2 (0.42) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL9456841 0.76 ABCC9 (0.73) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7349440 0.75 ABCC9 (0.58) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL9151647 0.74 NAMPT (0.51) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7357467 0.74 ABCC9 (0.57) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7348943 0.73 ABCC9 (0.54) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL7360174 0.72 NAMPT (0.50) ABCC9KCNJ11ABCC8KCNJ8CYP3A4
SCHEMBL11157791 0.71 ABCC9 (0.70) ABCC9KCNJ11ABCC8KCNJ8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP disclosed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US disclosed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO disclosed