SCHEMBL7347372

SCHEMBL7347372

CCOC(=O)C(CC)NC(=O)C1CC1C(=O)Nc1ccc(C=NN)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.37
TSHR P16473 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 3/20 0.35
NPC1 O15118 3/20 0.35
POLB P06746 2/20 0.35
ENPP3 O14638 1/20 0.35
ENPP1 P22413 1/20 0.35
ENPP2 Q13822 1/20 0.35
CAPN9 O14815 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
GAA P10253 1/20 0.34
AURKA O14965 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420630 0.88 KMT2A (0.39) RAB9ATSHRKMT2AALDH1A1NPC1
SCHEMBL9440351 0.84 RAB9A (0.37) RAB9ATSHRKMT2AALDH1A1NPC1
SCHEMBL9559149 0.81 LMNA (0.41) RAB9ATSHRKMT2AALDH1A1NPC1
SCHEMBL9558512 0.77 LMNA (0.43) RAB9ATSHRKMT2AALDH1A1NPC1
SCHEMBL9559156 0.76 MAPT (0.37) RAB9AKMT2AALDH1A1NPC1SMN1; SMN2
SCHEMBL6972945 0.76 PARP1 (0.49) RAB9ATSHRKMT2AALDH1A1NPC1
Hydrochloric Acid SCHEMBL7351854 0.75 PARP1 (0.48) RAB9ATSHRKMT2AALDH1A1NPC1
SCHEMBL7352508 0.73 ITGB3 (0.42) KMT2AALDH1A1POLBMAPTHPGD
SCHEMBL9559004 0.73 LMNA (0.42) RAB9ATSHRKMT2AALDH1A1MAPT
SCHEMBL9559001 0.73 LMNA (0.42) RAB9ATSHRKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542708-B1 Substituted beta-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2001-05-30 EP claimed
US-5973003-A TREATMENT OF THROMBOSIS, STROKE, MYOCARDIAL INFARCTION, INFLAMMATION AND ARTERIOSCLEROSIS G. D. SEARLE & CO. (US) 1999-10-26 US claimed
EP-0614360-B1 SUBSTITUTED BETA-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1997-03-19 EP claimed
EP-0542708-A1 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-05-19 EP claimed
US-5973003-A TREATMENT OF THROMBOSIS, STROKE, MYOCARDIAL INFARCTION, INFLAMMATION AND ARTERIOSCLEROSIS G. D. SEARLE & CO. (US) 1999-10-26 US disclosed
EP-0614360-B1 SUBSTITUTED BETA-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1997-03-19 EP disclosed
US-5344957-A Amidinoiphenyl-substituted G.D. SEARLE & CO. (US) 1994-09-06 US disclosed
EP-0542708-A1 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-05-19 EP disclosed
WO-1993007867-A1 SUBSTITUTED β-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-04-29 WO disclosed