SCHEMBL7347758

SCHEMBL7347758

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.52
CACNA1B Q00975 1/20 0.52
ADORA3 P0DMS8 3/20 0.52
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 5/20 0.51
HPGD P15428 4/20 0.51
CASP1 P29466 3/20 0.51
CASP7 P55210 3/20 0.51
HSD17B10 Q99714 3/20 0.51
GLA P06280 1/20 0.51
TSHR P16473 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CACNA1F O60840 1/20 0.48
CACNA1D Q01668 1/20 0.48
CACNA1S Q13698 1/20 0.48
CACNA1C Q13936 1/20 0.48
MAPT P10636 3/20 0.48
MAPK1 P28482 2/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367116 0.84 CACNA1B (0.50) GAACACNA1BADORA3ALDH1A1KDM4E
SCHEMBL7350838 0.83 HSD17B10 (0.63) GAACACNA1BADORA3ALDH1A1KDM4E
SCHEMBL7343709 0.83 CACNA1B (0.52) CACNA1BADORA3TSHRCACNA1FCACNA1D
SCHEMBL7349297 0.83 CACNA1B (0.57) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7341777 0.83 CACNA1F (0.63) ADORA3TSHRCACNA1FCACNA1DCACNA1S
SCHEMBL7345495 0.83 POLB (0.58) CACNA1BADORA3TSHRNPSR1CACNA1F
SCHEMBL7162019 0.83 GAA (0.63) GAACACNA1BADORA3ALDH1A1KDM4E
SCHEMBL7344603 0.83 KDM4E (0.67) GAAADORA3ALDH1A1KDM4EHPGD
SCHEMBL7344610 0.82 HSD17B10 (0.52) CACNA1BADORA3ALDH1A1KDM4EHPGD
SCHEMBL7343603 0.82 MAPT (0.70) ADORA3KDM4ETSHRNPSR1CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed