SCHEMBL7344610

SCHEMBL7344610

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1ccsc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 5/20 0.52
TSHR P16473 2/20 0.52
CACNA1B Q00975 1/20 0.52
ADORA3 P0DMS8 2/20 0.50
KDM4E B2RXH2 6/20 0.48
CASP1 P29466 3/20 0.48
HPGD P15428 3/20 0.48
PKM P14618 1/20 0.47
CACNA1F O60840 1/20 0.47
CACNA1D Q01668 1/20 0.47
CACNA1S Q13698 1/20 0.47
CACNA1C Q13936 1/20 0.47
ADORA2B P29275 3/20 0.46
ALDH1A1 P00352 3/20 0.46
CASP7 P55210 2/20 0.46
LMNA P02545 2/20 0.46
ADRA2A P08913 2/20 0.46
ADRA2B P18089 2/20 0.46
ADRA2C P18825 2/20 0.46
ADRA1D P25100 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10744164 0.83 ALDH1A1 (0.54) HSD17B10TSHRADORA3KDM4EHPGD
SCHEMBL7349611 0.83 HSD17B10 (0.64) HSD17B10TSHRCACNA1BADORA3KDM4E
SCHEMBL7341777 0.82 CACNA1F (0.63) TSHRADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7345495 0.82 POLB (0.58) TSHRCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL7343709 0.82 CACNA1B (0.52) TSHRCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL7347758 0.82 GAA (0.52) HSD17B10TSHRCACNA1BADORA3KDM4E
SCHEMBL7349297 0.82 CACNA1B (0.57) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7344613 0.81 ADORA3 (0.61) HSD17B10TSHRCACNA1BADORA3KDM4E
SCHEMBL7343547 0.80 ADORA3 (0.47) HSD17B10TSHRCACNA1BADORA3KDM4E
SCHEMBL7342397 0.80 ADORA3 (0.47) HSD17B10TSHRADORA3KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed