SCHEMBL7345495

SCHEMBL7345495

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1cccc(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.58
TSHR P16473 3/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CACNA1B Q00975 1/20 0.52
ADORA3 P0DMS8 4/20 0.52
MAPT P10636 5/20 0.51
CYP1A2 P05177 5/20 0.51
CYP3A4 P08684 5/20 0.51
CYP2C9 P11712 5/20 0.51
CYP2C19 P33261 5/20 0.51
ADRA1A P35348 4/20 0.51
CYP2D6 P10635 4/20 0.51
ABCB1 P08183 3/20 0.51
ADRA2A P08913 3/20 0.51
TDP1 Q9NUW8 3/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 2/20 0.51
ADRA1D P25100 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349297 0.89 CACNA1B (0.57) CACNA1BADORA3MAPTCYP1A2CYP3A4
SCHEMBL7341777 0.89 CACNA1F (0.63) POLBTSHRADORA3MAPTCYP1A2
SCHEMBL7343709 0.89 CACNA1B (0.52) POLBTSHRCACNA1BADORA3MAPT
SCHEMBL7349503 0.86 CACNA1C (0.65) POLBTSHRADORA3MAPTCYP1A2
SCHEMBL7343603 0.85 MAPT (0.70) POLBTSHRNPSR1ADORA3MAPT
SCHEMBL7343547 0.83 ADORA3 (0.47) TSHRNPSR1CACNA1BADORA3MAPT
SCHEMBL7340104 0.83 HSD17B10 (0.63) POLBTSHRNPSR1CACNA1BADORA3
SCHEMBL7347758 0.83 GAA (0.52) TSHRNPSR1CACNA1BADORA3MAPT
SCHEMBL7344610 0.82 HSD17B10 (0.52) POLBTSHRCACNA1BADORA3ADRA1A
SCHEMBL7345498 0.82 ADORA3 (0.64) POLBTSHRNPSR1CACNA1BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed