SCHEMBL7348455

SCHEMBL7348455

COc1cc(OCC(F)(F)F)c(F)cc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 5/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
RXRA P19793 1/20 0.41
HNF4A P41235 1/20 0.41
HSD17B10 Q99714 2/20 0.40
PYGL P06737 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3423769 0.82 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDLMNAMAPK1
SCHEMBL1487907 0.79 KDM4E (0.51) ALDH1A1KDM4ELMNAMAPK1HTT
SCHEMBL20107681 0.79 KDM4E (0.47) ALDH1A1KDM4EMAPK1CYP1A2CYP2C9
SCHEMBL7348451 0.78 KDM4E (0.42) ALDH1A1KDM4EHPGDLMNAMAPK1
SCHEMBL1931203 0.77 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDLMNAMAPK1
SCHEMBL15350432 0.77 CYP1A2 (0.54) ALDH1A1KDM4EHPGDMAPK1RAB9A
SCHEMBL3876532 0.77 CYP1A2 (0.61) ALDH1A1KDM4EHPGDMAPK1HTT
SCHEMBL5874056 0.74 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDLCKFYN
SCHEMBL2717570 0.74 POLB (0.41) ALDH1A1KDM4ECYP1A2CYP2C9RXRA
SCHEMBL20521864 0.74 KDM4E (0.51) ALDH1A1KDM4ELMNAMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726172-A BENZOXAZINONE DERIVATIVES; TREATMENT OF PRETERM LABOR, DYSMENORRHEA MERCK & CO., INC. (US) 1998-03-10 US disclosed
WO-1997025992-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-07-24 WO disclosed