SCHEMBL7348451

SCHEMBL7348451

COc1cc(OC(F)(F)CF)c(F)cc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.38
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
CTSV O60911 1/20 0.35
CTSL P07711 1/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
CD274 Q9NZQ7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3423769 0.81 ALDH1A1 (0.55) KDM4EALDH1A1HPGDLMNAHTT
SCHEMBL7348455 0.78 ALDH1A1 (0.43) KDM4EALDH1A1HPGDLMNAHTT
SCHEMBL1931203 0.76 ALDH1A1 (0.56) KDM4EALDH1A1HPGDLMNAHTT
SCHEMBL15462887 0.72 KDM4E (0.49) KDM4EALDH1A1HPGDLMNAHTT
SCHEMBL12444067 0.72 ALDH1A1 (0.64) KDM4EALDH1A1HPGDHTTLCK
SCHEMBL8595294 0.72 MAPT (0.35) KDM4E
SCHEMBL7349417 0.72 RAB9A (0.57) KDM4EALDH1A1LMNAHTTMAPK1
SCHEMBL2038394 0.72 KDM4E (0.40) KDM4EALDH1A1NPSR1KMT2A
SCHEMBL7349901 0.72 KDM4E (0.51) KDM4EALDH1A1HPGDLMNAHTT
SCHEMBL18713914 0.72 ALDH1A1 (0.51) KDM4EALDH1A1HPGDLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726172-A BENZOXAZINONE DERIVATIVES; TREATMENT OF PRETERM LABOR, DYSMENORRHEA MERCK & CO., INC. (US) 1998-03-10 US disclosed
WO-1997025992-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-07-24 WO disclosed