SCHEMBL7349147

SCHEMBL7349147

Cc1[nH]c(=O)[nH]c1C(=O)c1ccnc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.53
PDE4B Q07343 11/20 0.53
PDE4C Q08493 11/20 0.53
PDE4D Q08499 11/20 0.53
PDE3B Q13370 4/20 0.51
PDE3A Q14432 4/20 0.51
HPGD P15428 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
ATM Q13315 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HSD17B10 Q99714 1/20 0.51
BRAF P15056 1/20 0.39
TAS1R3 Q7RTX0 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430671 0.78 PDE3B (0.67) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL27623752 0.77 RECQL (0.47) TAS1R3TAS1R1TAS1R2SMARCA2SMARCA4
SCHEMBL11181578 0.76 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7340789 0.74 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20892726 0.73 LMNA (0.55) TAS1R3TAS1R1TAS1R2SMARCA2SMARCA4
SCHEMBL7339717 0.73 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7436668 0.72 LMNA (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7341027 0.72 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL5457930 0.71 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10635511 0.71 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169164-B1 IMIDAZOLONECARBONYLARYLIMIDAZOLES; METHOD OF MANUFACTURE, METHOD OF USE AND COMPOSITIONS USEFUL THEREOF SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-31 EP disclosed
US-4709043-A Process for the preparation of imidazolonecarbonylarylimidazoles SCHERING A.G. (DE) 1987-11-24 US disclosed
EP-0169164-A1 Imidazolonecarbonylarylimidazoles; method of manufacture, method of use and compositions useful thereof SCHERING AKTIENGESELLSCHAFT (DE) 1986-01-22 EP disclosed
US-4556665-A Cardiotonic 1,3-dihydro-4-[[(imidazol-1-yl)aryl]carbonyl]imidazol-2-ones SCHERING A.G. (DE) 1985-12-03 US disclosed