SCHEMBL7349554

SCHEMBL7349554

COc1ccc(S(=O)(=O)N(Cc2ccccc2)C(C(=O)OCc2ccccc2)C2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 2/20 0.65
MMP8 P22894 8/20 0.55
MMP13 P45452 8/20 0.55
MMP1 P03956 7/20 0.52
MMP3 P08254 7/20 0.52
MMP7 P09237 7/20 0.52
MMP9 P14780 7/20 0.52
MMP2 P08253 6/20 0.52
STS P08842 2/20 0.48
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
KMT2A Q03164 1/20 0.47
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
YAP1 P46937 1/20 0.45
GPR119 Q8TDV5 1/20 0.44
P2RX7 Q99572 2/20 0.44
TAS2R14 Q9NYV8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348074 1.00 BMP1 (0.65) BMP1MMP8MMP13MMP1MMP3
Hydrochloric Acid SCHEMBL7348358 0.99 BMP1 (0.64) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7354369 0.89 MMP13 (0.52) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7354374 0.87 MMP13 (0.53) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7354377 0.87 MMP13 (0.53) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7355697 0.84 BMP1 (0.59) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7355702 0.84 BMP1 (0.59) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7350312 0.83 TAS2R14 (0.48) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7350974 0.83 TAS2R14 (0.48) BMP1MMP8MMP13MMP1MMP3
SCHEMBL7350309 0.83 TAS2R14 (0.48) BMP1MMP8MMP13MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0766672-B1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS NOVARTIS AG (CH) 2000-10-04 EP disclosed
EP-0606046-B1 Arylsulfonamido-substituted hydroxamic acids CIBA GEIGY AG (CH) 1997-10-08 EP disclosed
US-5646167-A ADMINISTERED AS METALLOPROTEINASE INHIBITOR, ANTITUMOR OR ANTICARCINOGENIC AGENT CIBA-GEIGY CORPORATION (US) 1997-07-08 US disclosed
EP-0766672-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS Novartis AG (CH) 1997-04-09 EP disclosed
US-5552419-A METALLOPROTEINASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-09-03 US disclosed
US-5506242-A METALLOELASTASE INHIBITOR; TREATS EMPHYSEMA CIBA-GEIGY CORPORATION (US) 1996-04-09 US disclosed
WO-1996000214-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS CIBA-GEIGY AG (CH) 1996-01-04 WO disclosed
EP-0606046-A1 Arylsulfonamido-substituted hydroxamic acids CIBA-GEIGY AG (CH) 1994-07-13 EP disclosed