SCHEMBL7350256

SCHEMBL7350256

CCOC(=O)C1=C(C)NC(CSCNc2ccccc2)=C(C(=O)OCC)C1c1cccc(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 11/20 0.57
ADORA3 P0DMS8 2/20 0.50
ABCC1 P33527 1/20 0.47
CACNA1F O60840 2/20 0.46
CACNA1D Q01668 2/20 0.46
CACNA1S Q13698 2/20 0.46
CACNA1C Q13936 2/20 0.46
ACHE P22303 1/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
HIF1A Q16665 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7318265 0.89 CACNA1B (0.51) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL7322259 0.88 CACNA1B (0.53) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL9501260 0.86 ADORA3 (0.57) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL7316147 0.85 ADORA3 (0.53) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7419122 0.83 ADORA3 (0.53) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL7266098 0.82 CACNA1B (0.51) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL9808332 0.81 ABCC1 (0.48) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL7471880 0.80 ADORA3 (0.51) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL9513394 0.80 ABCC1 (0.58) CACNA1BADORA3ABCC1CACNA1FCACNA1D
SCHEMBL11522715 0.80 ABCC1 (0.58) CACNA1BADORA3ABCC1CACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0271059-B1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA (IT) 1993-10-20 EP claimed
EP-0271059-A1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1988-06-15 EP claimed