SCHEMBL7350845

SCHEMBL7350845

COc1ccc(S(=O)(=O)N(CCN2CCOCC2)CC(=O)NO)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 6/20 1.00
BMP1 P13497 3/20 0.83
MMP1 P03956 3/20 0.65
MMP13 P45452 3/20 0.65
MMP7 P09237 2/20 0.65
MMP8 P22894 2/20 0.65
MMP12 P39900 2/20 0.65
MEP1B Q16820 3/20 0.64
ALDH1A1 P00352 4/20 0.63
GAA P10253 1/20 0.57
MMP9 P14780 1/20 0.52
ADAM17 P78536 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004503 0.91 BMP1 (1.00) MMP3BMP1MMP1MMP13MMP7
SCHEMBL7346814 0.89 MMP3 (1.00) MMP3BMP1MMP1MMP13MMP7
SCHEMBL6626956 0.86 MMP3 (0.75) MMP3BMP1MMP1MMP13MMP7
Hydrochloric Acid SCHEMBL3938385 0.85 MMP3 (0.73) MMP3BMP1MMP1MMP13MMP7
SCHEMBL7341155 0.84 MMP3 (0.73) MMP3BMP1MMP1MMP13ALDH1A1
SCHEMBL7451485 0.84 MMP3 (0.73) MMP3BMP1MMP1MMP13MMP7
SCHEMBL6794166 0.82 MMP3 (0.69) MMP3BMP1MMP1MMP13MMP7
SCHEMBL26776688 0.80 MMP1 (0.81) MMP3BMP1MMP1MMP13MMP7
SCHEMBL26776708 0.79 MMP1 (0.79) MMP3BMP1MMP1MMP13MMP7
SCHEMBL6804953 0.79 MMP3 (0.65) MMP3BMP1MMP1MMP13MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0766672-B1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS NOVARTIS AG (CH) 2000-10-04 EP disclosed
EP-0606046-B1 Arylsulfonamido-substituted hydroxamic acids CIBA GEIGY AG (CH) 1997-10-08 EP disclosed
US-5646167-A ADMINISTERED AS METALLOPROTEINASE INHIBITOR, ANTITUMOR OR ANTICARCINOGENIC AGENT CIBA-GEIGY CORPORATION (US) 1997-07-08 US disclosed
EP-0766672-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS Novartis AG (CH) 1997-04-09 EP disclosed
WO-1996040101-A1 CERTAIN ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS FOR THE TREATMENT OF CERTAIN TUMORS NOVARTIS AG (CH) 1996-12-19 WO disclosed
US-5552419-A METALLOPROTEINASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-09-03 US disclosed
US-5506242-A METALLOELASTASE INHIBITOR; TREATS EMPHYSEMA CIBA-GEIGY CORPORATION (US) 1996-04-09 US disclosed
WO-1996000214-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS CIBA-GEIGY AG (CH) 1996-01-04 WO disclosed
US-5455258-A Useful as inhibitors of matrix-degrading metalloproteinase enzymes such as stromelysin and/or collegenase CIBA-GEIGY CORPORATION (US) 1995-10-03 US disclosed
EP-0606046-A1 Arylsulfonamido-substituted hydroxamic acids CIBA-GEIGY AG (CH) 1994-07-13 EP disclosed