SCHEMBL7350857

SCHEMBL7350857

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCc2cc(C)[nH]c2C)C1c1cccc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.57
CACNA1B Q00975 1/20 0.51
ADORA3 P0DMS8 1/20 0.50
CACNA1F O60840 5/20 0.49
CACNA1D Q01668 5/20 0.49
CACNA1S Q13698 5/20 0.49
CACNA1C Q13936 5/20 0.49
HIF1A Q16665 3/20 0.49
MEN1 O00255 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
KMT2A Q03164 2/20 0.49
MAPT P10636 2/20 0.49
TSHR P16473 2/20 0.49
LMNA P02545 1/20 0.49
MAPK1 P28482 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344543 0.89 CACNA1B (0.52) POLBCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL7338912 0.89 CACNA1B (0.55) POLBCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL7344807 0.89 CACNA1F (0.64) POLBADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7344759 0.86 CACNA1F (0.66) POLBADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7350545 0.85 MEN1 (0.71) POLBADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7350085 0.84 ALDH1A1 (0.53) POLBCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL7343213 0.83 ADORA3 (0.46) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL3024959 0.83 CACNA1B (0.62) POLBCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL3326231 0.82 TSHR (0.69) POLBCACNA1BADORA3CACNA1FCACNA1D
SCHEMBL29676320 0.82 TSHR (0.69) POLBCACNA1BADORA3CACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed