SCHEMBL7353282

SCHEMBL7353282

CCOP(=O)(CCCn1c(=O)c(=O)[nH]c2cc([N+](=O)[O-])ccc21)OCC

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.45
SIRT1 Q96EB6 1/20 0.45
GRIK1 P39086 2/20 0.42
GRIK2 Q13002 2/20 0.42
GRIK3 Q13003 2/20 0.42
GRIK4 Q16099 2/20 0.42
GRIK5 Q16478 2/20 0.42
GRIA1 P42261 1/20 0.40
GRIA2 P42262 1/20 0.40
GRIA3 P42263 1/20 0.40
GRIA4 P48058 1/20 0.40
CYP1A2 P05177 1/20 0.39
PARP1 P09874 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354078 0.87 SIRT2 (0.43) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7361295 0.84 SIRT2 (0.46) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7358401 0.81 GRIA1 (0.45) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL9542780 0.81 SIRT2 (0.52) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7354618 0.81 SIRT2 (0.46) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7353289 0.81 GRIK1 (0.40) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7353360 0.80 GRIK1 (0.59) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL7357748 0.79 SIRT2 (0.48) SIRT2SIRT1GRIK1GRIK2GRIK3
SCHEMBL8609548 0.79 CYP1A2 (0.57) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7353149 0.78 PARG (0.42) SIRT2SIRT1GRIK1GRIK2GRIK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed