SCHEMBL9542780

SCHEMBL9542780

CCCn1c(=O)c(=O)[nH]c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.52
SIRT1 Q96EB6 1/20 0.52
GRIA1 P42261 1/20 0.50
GRIA2 P42262 1/20 0.50
GRIA3 P42263 1/20 0.50
GRIA4 P48058 1/20 0.50
CYP1A2 P05177 1/20 0.48
PARP1 P09874 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
CFTR P13569 1/20 0.46
GRIK1 P39086 2/20 0.44
GRIK2 Q13002 2/20 0.44
GRIK3 Q13003 2/20 0.44
GRIK4 Q16099 2/20 0.44
GRIK5 Q16478 2/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MPI P34949 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8609548 0.89 CYP1A2 (0.57) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7349770 0.85 GRIK1 (0.61) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7357748 0.83 SIRT2 (0.48) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7361791 0.82 GRIA1 (0.48) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL9395642 0.82 GRIA1 (0.57) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL31439102 0.82 GRIA1 (0.57) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL31439101 0.82 GRIA1 (0.57) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7355281 0.82 GRIK1 (0.55) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7353360 0.81 GRIK1 (0.59) SIRT2SIRT1GRIA1GRIA2GRIA3
SCHEMBL7353282 0.81 SIRT2 (0.45) SIRT2SIRT1GRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993008173-A1 QUINOXALINE DERIVATES WITH AFFINITY FOR QUISQUALATE-RECEPTORS SCHERING AKTIENGESELLSCHAFT (DE) 1993-04-29 WO disclosed