SCHEMBL7354047

SCHEMBL7354047

O=C(O)Cc1ccc(Cn2c(=O)c(=O)n(Cc3ccc(C(=O)O)cc3)c3ccc([N+](=O)[O-])cc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.47
SRC P12931 2/20 0.46
PRKACA P17612 1/20 0.46
PRKACG P22612 1/20 0.46
PRKACB P22694 1/20 0.46
NOX4 Q9NPH5 1/20 0.46
CYP1A2 P05177 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
POLB P06746 1/20 0.44
IDO1 P14902 1/20 0.43
PLA2G2A P14555 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MITF O75030 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
DCTPP1 Q9H773 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356210 0.81 TP53 (0.52) CCR2NOX4CYP1A2KMT2AMEN1
SCHEMBL7352345 0.81 CCR2 (0.46) CCR2SRCPRKACAPRKACGPRKACB
SCHEMBL7361149 0.81 SMN1; SMN2 (0.51) SRCPRKACAPRKACGPRKACBNOX4
SCHEMBL7352784 0.79 PGR (0.49) CCR2SRCPRKACAPRKACGPRKACB
SCHEMBL7361866 0.75 CFTR (0.48) CCR2NOX4KMT2AMEN1PLA2G2A
SCHEMBL7354439 0.73 CYP1A2 (0.48) NOX4CYP1A2TDP1KMT2AMEN1
SCHEMBL3192269 0.71 PPARG (0.54) CCR2TDP1
SCHEMBL18180381 0.71 CYP1A2 (0.66) CCR2CYP1A2POLBMAPT
SCHEMBL30643815 0.71 CYP2C19 (0.64) CYP1A2TDP1KMT2AMEN1IDO1
SCHEMBL76204 0.71 CYP2C19 (0.64) CYP1A2TDP1KMT2AMEN1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed