SCHEMBL7354598

SCHEMBL7354598

NC(=O)CCC(=O)NCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.64
LMNA P02545 1/20 0.64
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
TPSAB1 Q15661 2/20 0.57
GAA P10253 1/20 0.57
TRPV1 Q8NER1 2/20 0.55
EPHX2 P34913 1/20 0.53
NR1H4 Q96RI1 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HTT P42858 2/20 0.51
HDAC1 Q13547 3/20 0.51
AOC3 Q16853 2/20 0.51
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4900724 0.90 GAA (0.70) ALDH1A1MEN1KMT2ATPSAB1GAA
SCHEMBL8245493 0.84 LMNA (0.64) ALDH1A1LMNAMEN1KMT2AGAA
SCHEMBL7348903 0.84 SRC (0.57) ALDH1A1LMNATPSAB1HTTAOC3
SCHEMBL10031020 0.83 MEN1 (0.80) ALDH1A1LMNAMEN1KMT2ATPSAB1
SCHEMBL7350032 0.83 LTB4R2 (0.52) ALDH1A1LMNAMEN1KMT2ATPSAB1
SCHEMBL7352930 0.83 MME (0.52) ALDH1A1LMNAMEN1KMT2ATPSAB1
SCHEMBL8792470 0.82 ALDH1A1 (0.71) ALDH1A1LMNAMEN1KMT2AGAA
SCHEMBL7351961 0.82 TPSAB1 (0.51) ALDH1A1LMNAMEN1KMT2ATPSAB1
SCHEMBL13073870 0.81 AOC3 (0.73) ALDH1A1LMNAMEN1KMT2ATPSAB1
SCHEMBL27703735 0.81 MEN1 (0.83) ALDH1A1LMNAMEN1KMT2ATPSAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005448-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS Du Pont Pharmaceuticals Company (US) 2000-06-07 EP claimed
WO-1999009000-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS DU PONT PHARMACEUTICALS COMPANY (US) 1999-02-25 WO claimed
EP-1005448-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS Du Pont Pharmaceuticals Company (US) 2000-06-07 EP disclosed
WO-1999009000-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS DU PONT PHARMACEUTICALS COMPANY (US) 1999-02-25 WO disclosed