SCHEMBL7354869

SCHEMBL7354869

N#C/N=C(\Nc1cccnc1)NC1(c2ccccc2)CC=CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
KMT2A Q03164 3/20 0.40
PKM P14618 1/20 0.40
MEN1 O00255 1/20 0.40
ABCC9 O60706 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
ABCC8 Q09428 1/20 0.40
KCNJ11 Q14654 1/20 0.40
KCNJ8 Q15842 1/20 0.40
LMNA P02545 2/20 0.40
NAMPT P43490 4/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 2/20 0.38
GRIN2B Q13224 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354870 1.00 P2RX7 (0.41) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL13949288 0.91 P2RX7 (0.43) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL4264238 0.91 P2RX7 (0.43) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL13949283 0.89 P2RX7 (0.41) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL7357917 0.89 P2RX7 (0.41) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL4259491 0.89 P2RX7 (0.41) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL11156357 0.80 RAB9A (0.57) P2RX7NPC1RAB9AKMT2APKM
SCHEMBL7348975 0.77 ALDH1A1 (0.43) P2RX7NPC1KMT2APKMMEN1
SCHEMBL7348973 0.77 ALDH1A1 (0.43) P2RX7NPC1KMT2APKMMEN1
SCHEMBL7360161 0.76 P2RX7 (0.43) P2RX7NPC1RAB9AKMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP disclosed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US disclosed
EP-0655057-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS. UPJOHN CO (US) 1995-05-31 EP disclosed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO disclosed