SCHEMBL7355425

SCHEMBL7355425

CC(Cc1ccccc1F)NC(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 17/20 0.57
METAP1 P53582 9/20 0.57
DPP4 P27487 2/20 0.40
FAP Q12884 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7360183 0.99 METAP2 (0.56) METAP2METAP1DPP4FAPDPP8
SCHEMBL14984955 0.87 METAP2 (0.44) METAP2METAP1DPP4FAPDPP8
SCHEMBL12022087 0.86 METAP2 (0.43) METAP2METAP1DPP4FAPDPP8
SCHEMBL21928685 0.86 METAP2 (0.43) METAP2METAP1DPP4FAPDPP8
SCHEMBL7362423 0.82 METAP2 (0.63) METAP2METAP1
Hydrochloric Acid SCHEMBL7352923 0.81 METAP2 (0.62) METAP2METAP1
SCHEMBL7360854 0.81 METAP2 (0.60) METAP2METAP1ALDH1A1
Hydrochloric Acid SCHEMBL7349814 0.80 METAP2 (0.58) METAP2METAP1ALDH1A1
SCHEMBL23710451 0.78 METAP2 (0.38) METAP2METAP1DPP4FAPDPP8
SCHEMBL6477759 0.78 METAP2 (0.72) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed