SCHEMBL7355758

SCHEMBL7355758

CCCCCc1cc(OS(=O)(=O)C(F)(F)F)c2occc2c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41
FUT7 Q11130 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
DRD2 P14416 2/20 0.33
DRD1 P21728 2/20 0.33
DRD4 P21917 2/20 0.33
DRD5 P21918 2/20 0.33
DRD3 P35462 2/20 0.33
KCNH2 Q12809 5/20 0.33
CA12 O43570 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352238 0.80 CYP3A4 (0.36) CA2CA1CA9PPARGDRD2
SCHEMBL7940562 0.79 CYP3A4 (0.31)
SCHEMBL7350220 0.79 CYP3A4 (0.31)
SCHEMBL7351472 0.79 DRD2 (0.34) CA2CA1PPARGPPARADRD2
SCHEMBL7940582 0.79 PPARG (0.45) PPARGPPARACNR1CNR2
SCHEMBL10179904 0.74 CA2 (0.62) CA2CA1CA9FUT7TRPV1
SCHEMBL18351666 0.73 PPARA (0.41) CA2CA1CA9FUT7PPARG
SCHEMBL9698561 0.73 FUT7 (0.45) CA2CA1CA9FUT7PPARG
SCHEMBL10455918 0.73 PPARG (0.42) CA2CA1CA9PPARGPPARA
SCHEMBL20048158 0.73 PPARA (0.42) CA2CA1CA9FUT7PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0834508-B1 Substituted biphenyl or phenylpyridine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-08-16 EP disclosed
EP-1009736-A1 MALONIC ACID BASED MATRIX METALLOPROTEINASE INHIBITORS Roche Diagnostics GmbH (DE) 2000-06-21 EP disclosed
WO-1999011608-A1 MALONIC ACID BASED MATRIX METALLOPROTEINASE INHIBITORS ROCHE DIAGNOSTICS GMBH (DE) 1999-03-11 WO disclosed
EP-0834508-A1 Substituted biphenyl or phenylpyridine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-04-08 EP disclosed