SCHEMBL7356104

SCHEMBL7356104

COc1cc(-c2nc3ccc(C4(C)C=NNC(=O)C4)cc3[nH]2)cc(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
BLM P54132 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
AMY1A P0DUB6 8/20 0.42
ALOX5 P09917 1/20 0.41
EPHX2 P34913 1/20 0.41
CDKN1A P38936 3/20 0.39
PARP1 P09874 1/20 0.39
KDR P35968 1/20 0.39
ABCB11 O95342 1/20 0.38
MAOA P21397 1/20 0.38
ADORA2A P29274 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357077 0.86 ABCB11 (0.52) KDM4EMEN1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL11304721 0.85 ABCB11 (0.52) KDM4EMEN1ALDH1A1GAAMAPT
SCHEMBL7350293 0.83 NPC1 (0.49) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL11306274 0.83 AMY1A (0.43) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL7352293 0.83 NPC1 (0.49) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL11302741 0.83 NPBWR1 (0.48) KDM4EMEN1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL11307551 0.82 AMY1A (0.42) KDM4EMEN1ALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL11302544 0.82 NPC1 (0.48) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL7355829 0.82 MEN1 (0.48) KDM4EMEN1ALDH1A1GAAMAPT
SCHEMBL8891480 0.82 SCD (0.50) ALDH1A1SMN1; SMN2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361563-A CARDIOTONIC, ANTITHROMBOTIC DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-11-30 US disclosed
EP-0008391-A1 Benzimidazoles, their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1980-03-05 EP disclosed