SCHEMBL7356239

SCHEMBL7356239

CCOC(=O)Cn1c(C)cc(Cl)c([N+](=O)[O-])c1=O

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 3/20 0.47
RAB9A P51151 2/20 0.44
TSHR P16473 1/20 0.43
APOBEC3A P31941 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
MITF O75030 1/20 0.41
ENPP2 Q13822 1/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356005 0.80 ALDH1A1 (0.42) ALDH1A1KDM4ERAB9ATSHRMITF
SCHEMBL7364209 0.79 ALDH1A1 (0.41) ALDH1A1KDM4ERAB9ATSHRMITF
SCHEMBL7356994 0.79 ALDH1A1 (0.42) ALDH1A1KDM4ERAB9ATSHRMITF
SCHEMBL8030820 0.77 MITF (0.47) ALDH1A1KDM4ERAB9AMITFLMNA
SCHEMBL7360418 0.76 MITF (0.46) ALDH1A1KDM4ERAB9AMITFLMNA
SCHEMBL7360414 0.75 MITF (0.45) ALDH1A1KDM4ERAB9AMITFLMNA
SCHEMBL7773566 0.74 MAPT (0.44) ALDH1A1KDM4ERAB9ATSHRSMN1; SMN2
Propane SCHEMBL8025594 0.73 ALDH1A1 (0.39) ALDH1A1RAB9ATSHRMITFLMNA
SCHEMBL7771930 0.72 SMN1; SMN2 (0.43) ALDH1A1KDM4ERAB9ATSHRMITF
SCHEMBL13120802 0.70 ALDH1A1 (0.44) ALDH1A1KDM4ERAB9AMITFLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117660-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-01-09 EP disclosed
EP-1117660-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2001-07-25 EP disclosed
US-6117888-A N-((2-AMINO-6-METHYLPYRID-5YL)METHYLAMINOCARBONYLMETHYL)PYRIDO NE-4-SULFONAMIDES MERCK & CO., INC. (US) 2000-09-12 US disclosed
WO-2000018762-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2000-04-06 WO disclosed