SCHEMBL7356445

SCHEMBL7356445

O=[N+]([O-])c1ccc(S(=O)(=O)CCCCCO)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.60
GSTP1 P09211 1/20 0.49
TSHR P16473 1/20 0.47
HSD11B1 P28845 1/20 0.47
CA1 P00915 5/20 0.46
MMP1 P03956 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
CA12 O43570 4/20 0.46
CA9 Q16790 4/20 0.46
CA14 Q9ULX7 4/20 0.46
CA3 P07451 3/20 0.46
CA4 P22748 3/20 0.46
CA6 P23280 3/20 0.46
CA5A P35218 3/20 0.46
CA7 P43166 3/20 0.46
CA13 Q8N1Q1 3/20 0.46
CA5B Q9Y2D0 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340091 0.86 CA2 (0.58) CA2TSHRHSD11B1CA1MMP1
SCHEMBL7356440 0.85 CA2 (0.47) CA2HSD11B1CA1MMP1MMP2
SCHEMBL11309979 0.84 CA2 (0.81) CA2GSTP1MMP1MMP8MMP13
SCHEMBL7538187 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14
SCHEMBL20468019 0.83 CA2 (0.50) CA2HSD11B1CA1MMP1MMP2
SCHEMBL11134832 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14
SCHEMBL17603652 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14
SCHEMBL30426244 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14
SCHEMBL7537992 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14
SCHEMBL7541961 0.83 ALDH1A1 (0.56) CA2CA1CA12CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed