SCHEMBL73586

SCHEMBL73586

CCOC(=O)Cc1cc(Cl)c(NC(=O)c2csc3ccccc23)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.45
TP53 P04637 3/20 0.45
RAB9A P51151 3/20 0.45
MEN1 O00255 3/20 0.45
MAPT P10636 3/20 0.45
KMT2A Q03164 3/20 0.45
NPC1 O15118 2/20 0.45
NFKB1 P19838 2/20 0.45
HTT P42858 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
HSD17B10 Q99714 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
NFATC1 O95644 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70894 0.88 PIK3CA (0.46) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL72046 0.85 PTGDR2 (0.51) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL5708317 0.82 SMN1; SMN2 (0.43) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL72217 0.79 MAPT (0.41) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL5161089 0.73 HDAC3 (0.51) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL73096 0.72 PTGDR2 (0.52) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL91763 0.71 RAB9A (0.64) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL91757 0.71 HDAC3 (0.52) SMN1; SMN2TP53RAB9AMEN1MAPT
SCHEMBL8787255 0.70 SMN1; SMN2 (0.56) SMN1; SMN2TP53MEN1MAPTKMT2A
SCHEMBL9494725 0.70 TSHR (0.58) SMN1; SMN2TP53RAB9AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed