SCHEMBL70894

SCHEMBL70894

CCOC(=O)Cc1ccc(NC(=O)c2csc3ccccc23)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.45
RAB9A P51151 5/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
NPC1 O15118 3/20 0.43
NFKB1 P19838 3/20 0.43
NFKB2 Q00653 3/20 0.43
RELA Q04206 3/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 2/20 0.43
HTT P42858 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MCOLN3 Q8TDD5 1/20 0.43
NFATC1 O95644 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL73586 0.88 SMN1; SMN2 (0.45) PIK3CAPTGDR2RAB9ASMN1; SMN2NPC1
SCHEMBL5708317 0.86 SMN1; SMN2 (0.43) PIK3CAPTGDR2RAB9ASMN1; SMN2NPC1
SCHEMBL73096 0.85 PTGDR2 (0.52) PIK3CAPTGDR2RAB9ASMN1; SMN2NPC1
SCHEMBL72217 0.83 MAPT (0.41) PIK3CAPTGDR2RAB9ASMN1; SMN2NPC1
SCHEMBL91763 0.81 RAB9A (0.64) RAB9ASMN1; SMN2NPC1NFKB1NFKB2
SCHEMBL2438042 0.80 ITGB1 (0.53) PTGDR2RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL2429129 0.79 ITGB1 (0.55) RAB9AMAPTKMT2ANPSR1HDAC1
SCHEMBL91757 0.76 HDAC3 (0.52) PIK3CARAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL13566602 0.76 SGMS2 (0.52) RAB9ASMN1; SMN2NPC1MAPTTP53
SCHEMBL14491729 0.76 POLB (0.45) RAB9ASMN1; SMN2NPC1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed