SCHEMBL7359494

SCHEMBL7359494

O=C1N(CCC2CCN(CC3COc4ccccc4O3)CC2)CCCN1c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.55
SIGMAR1 Q99720 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17272740 0.88 HTR1A (0.52) HTR1ASIGMAR1
SCHEMBL17272705 0.83 HTR1A (0.56) HTR1ASIGMAR1
SCHEMBL7437505 0.83 HTR1A (0.47) HTR1ASIGMAR1
SCHEMBL17272733 0.83 HTR1A (0.57) HTR1ASIGMAR1
SCHEMBL15865440 0.82 HTR1A (0.63) HTR1ASIGMAR1
SCHEMBL7430039 0.81 HTR1A (0.51) HTR1ASIGMAR1
SCHEMBL15870257 0.80 HTR1A (0.58) HTR1ASIGMAR1
SCHEMBL17272720 0.80 HTR1A (0.58) HTR1ASIGMAR1
SCHEMBL15865438 0.80 HTR1A (0.58) HTR1ASIGMAR1
SCHEMBL7366546 0.79 SIGMAR1 (0.62) HTR1ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997028157-A1 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed