SCHEMBL7366546

SCHEMBL7366546

O=C1CC(CN2CCC(CCN3CCN(c4ccccc4)C3=O)CC2)Oc2ccccc21

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.62
HTR1A P08908 1/20 0.62
ABCB1 P08183 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359494 0.79 HTR1A (0.55) SIGMAR1HTR1A
SCHEMBL7366544 0.78 SIGMAR1 (0.61) SIGMAR1HTR1AABCB1
SCHEMBL17272740 0.78 HTR1A (0.52) SIGMAR1HTR1A
SCHEMBL7365851 0.74 ACHE (0.62)
SCHEMBL7437505 0.74 HTR1A (0.47) SIGMAR1HTR1A
SCHEMBL7365661 0.72 DRD2 (0.43)
SCHEMBL7430039 0.72 HTR1A (0.51) SIGMAR1HTR1A
SCHEMBL17272733 0.71 HTR1A (0.57) SIGMAR1HTR1A
SCHEMBL7367467 0.71 DRD2 (0.57)
SCHEMBL15865440 0.71 HTR1A (0.63) SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997028157-A1 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed