SCHEMBL7359563

SCHEMBL7359563

CCC(c1ccccc1)c1c(O)c2ccc(OCCOCCOC)cc2oc1=O

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 8/20 0.58
NQO1 P15559 1/20 0.47
VKORC1 Q9BQB6 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
ALB P02768 1/20 0.45
PCSK7 Q16549 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ACHE P22303 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359481 0.86 CYP2C9 (0.67) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7354536 0.85 CYP2C9 (0.69) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL27418866 0.82 CYP2C9 (0.61) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7354675 0.80 CCR4 (0.54) CYP2C9ACHE
SCHEMBL7400115 0.79 ACHE (0.40) CYP2C9NQO1VKORC1ACHE
SCHEMBL7357584 0.78 CYP2C9 (0.76) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL9211359 0.77 ACHE (0.56) NQO1KDM4EALDH1A1MEN1KMT2A
SCHEMBL7355347 0.77 CYP2C9 (0.74) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7352607 0.76 CYP2C9 (0.69) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7359848 0.76 CYP2C9 (0.72) CYP2C9NQO1VKORC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682663-B1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS UPJOHN CO (US) 2001-04-18 EP claimed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US claimed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP claimed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO claimed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP disclosed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO disclosed