SCHEMBL7360649

SCHEMBL7360649

COC(=O)C=CCN(CCc1ccc([N+](=O)[O-])cc1)c1cccc(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.44
KCNJ1 P48048 2/20 0.44
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
NLRP1 Q9C000 1/20 0.38
P4HB P07237 1/20 0.38
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
THRB P10828 1/20 0.37
APEX1 P27695 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458452 1.00 KCNH2 (0.44) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL7361984 0.89 FFAR1 (0.40) MEN1KMT2AALDH1A1MAPTP4HB
SCHEMBL7361986 0.89 FFAR1 (0.40) MEN1KMT2AALDH1A1MAPTP4HB
SCHEMBL7362625 0.78 KCNH2 (0.46) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL7363729 0.72 KCNH2 (0.50) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL7360601 0.72 KCNH2 (0.44) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL7363865 0.72 KCNH2 (0.47) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL7462970 0.72 KCNH2 (0.43) KCNH2KCNJ1ALDH1A1MAPTMAOA
SCHEMBL7362630 0.71 KCNH2 (0.47) KCNH2KCNJ1CDC25C
SCHEMBL7368633 0.71 NR1H4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed