SCHEMBL7363729

SCHEMBL7363729

N#Cc1cccc(N(CCCO)CCCCc2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.50
KCNJ1 P48048 2/20 0.50
TSHR P16473 1/20 0.44
SLC22A2 O15244 1/20 0.40
ADRB1 P08588 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC47A2 Q86VL8 1/20 0.40
SLC47A1 Q96FL8 1/20 0.40
FFAR1 O14842 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
FBP1 P09467 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7363865 0.86 KCNH2 (0.47) KCNH2KCNJ1TSHRFFAR1MEN1
SCHEMBL7360601 0.82 KCNH2 (0.44) KCNH2KCNJ1MEN1KMT2AALDH1A1
SCHEMBL8345485 0.82 KCNH2 (0.47) KCNH2KCNJ1TSHRFFAR1MEN1
SCHEMBL7365992 0.79 KCNH2 (0.46) KCNH2KCNJ1FFAR1ALDH1A1CA12
SCHEMBL7360603 0.77 KCNH2 (0.45) KCNH2KCNJ1FFAR1ALDH1A1CA12
SCHEMBL7462980 0.76 KCNH2 (0.44) KCNH2KCNJ1SLC22A2ADRB1SLC6A4
SCHEMBL2418609 0.76 ALDH1A1 (0.54) TSHRMEN1KMT2AALDH1A1POLB
SCHEMBL7462970 0.76 KCNH2 (0.43) KCNH2KCNJ1SLC22A2ADRB1SLC6A4
SCHEMBL7457058 0.75 KCNJ1 (0.54) KCNH2KCNJ1TSHRMEN1KMT2A
SCHEMBL8350250 0.74 KCNH2 (0.46) KCNH2KCNJ1FFAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed