SCHEMBL7361087

SCHEMBL7361087

NC(=O)C1(C[CH]C(=O)NCC(=O)c2oc(-c3cccnc3)nc2CC2CCCCC2)CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.34
KCNH2 Q12809 1/20 0.34
ATM Q13315 1/20 0.34
ATR Q13535 1/20 0.34
IKBKB O14920 1/20 0.34
ALDH1A1 P00352 2/20 0.33
GAA P10253 1/20 0.33
BMP1 P13497 1/20 0.32
NAMPT P43490 1/20 0.32
GBA1 P04062 1/20 0.32
TP53 P04637 1/20 0.31
FPR2 P25090 1/20 0.31
LMNA P02545 1/20 0.31
USP2 O75604 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806965 0.84 RAB9A (0.38) RAB9AKCNH2ATMATRIKBKB
SCHEMBL7361089 0.80 IKBKB (0.39) RAB9AKCNH2ATMATRIKBKB
SCHEMBL6802384 0.80 BMP1 (0.38) RAB9AKCNH2ATMATRIKBKB
SCHEMBL6798235 0.78 RAB9A (0.36) RAB9AKCNH2ATMATRIKBKB
SCHEMBL7357734 0.78 RAB9A (0.39) RAB9AKCNH2ATMATRIKBKB
SCHEMBL6806971 0.78 AAK1 (0.43) RAB9AKCNH2ATMATRIKBKB
SCHEMBL6802381 0.73 CNR1 (0.37) TP53LMNA
SCHEMBL6798242 0.72 RAB9A (0.39) RAB9AKCNH2ATMATRALDH1A1
SCHEMBL6800322 0.69 KDM4E (0.38) RAB9AIKBKBALDH1A1TP53MKNK1
SCHEMBL6803048 0.65 RAB9A (0.36) RAB9AIKBKBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed