SCHEMBL7361089

SCHEMBL7361089

NC(=O)C(C(=O)NCC(=O)c1oc(-c2cccnc2)nc1CC1CCCCC1)C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.39
RAB9A P51151 1/20 0.39
BMP1 P13497 1/20 0.37
ATM Q13315 2/20 0.37
ATR Q13535 2/20 0.37
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
GBA1 P04062 1/20 0.34
MMP13 P45452 1/20 0.34
REN P00797 1/20 0.33
PTGES O14684 2/20 0.33
EGLN1 Q9GZT9 1/20 0.33
DHPS P49366 1/20 0.33
FPR2 P25090 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802384 0.86 BMP1 (0.38) IKBKBRAB9ABMP1ATMATR
SCHEMBL6806971 0.84 AAK1 (0.43) IKBKBRAB9ABMP1ATMATR
SCHEMBL6806965 0.83 RAB9A (0.38) IKBKBRAB9ABMP1ATMATR
SCHEMBL7357734 0.83 RAB9A (0.39) IKBKBRAB9ABMP1ATMATR
SCHEMBL7361087 0.80 RAB9A (0.34) IKBKBRAB9ABMP1ATMATR
SCHEMBL6798242 0.78 RAB9A (0.39) RAB9ABMP1ATMATRKCNH2
SCHEMBL6798235 0.77 RAB9A (0.36) IKBKBRAB9ABMP1ATMATR
SCHEMBL6800330 0.70 AAK1 (0.45) IKBKBRAB9AALDH1A1
SCHEMBL6802381 0.69 CNR1 (0.37) LMNA
SCHEMBL6800014 0.68 SMN1; SMN2 (0.38) RAB9ABMP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed