SCHEMBL7361301

SCHEMBL7361301

O=C(C=C(O)C(F)(F)F)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.57
ALDH1A1 P00352 5/20 0.56
CES1 P23141 2/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
MAPK1 P28482 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HDAC3 O15379 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
AKT1 P31749 1/20 0.48
MAOB P27338 2/20 0.44
CYP1B1 Q16678 2/20 0.44
RECQL P46063 2/20 0.44
MAPT P10636 2/20 0.44
LMNA P02545 2/20 0.44
PLIN1 O60240 1/20 0.44
BCHE P06276 1/20 0.44
TNFRSF1A P19438 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361299 1.00 NFE2L2 (0.57) NFE2L2ALDH1A1CES1MEN1KMT2A
SCHEMBL12900918 1.00 NFE2L2 (0.57) NFE2L2ALDH1A1CES1MEN1KMT2A
SCHEMBL23978379 0.88 NFE2L2 (0.57) NFE2L2ALDH1A1CES1MEN1KMT2A
SCHEMBL29116567 0.83 NFE2L2 (0.57) NFE2L2ALDH1A1CES1MEN1KMT2A
SCHEMBL2704264 0.82 ALDH1A1 (0.59) ALDH1A1CES1MEN1KMT2AMAOB
SCHEMBL5308087 0.82 CYP1B1 (0.46) ALDH1A1CES1MEN1KMT2ATDP1
SCHEMBL6029412 0.82 NR4A1 (0.54) CES1MAOBCYP1B1CYP1A1CES2
SCHEMBL2704266 0.82 ALDH1A1 (0.59) ALDH1A1CES1MEN1KMT2AMAOB
SCHEMBL25341875 0.82 PLOD2 (0.47) NFE2L2ALDH1A1MEN1KMT2AMAPK1
SCHEMBL5308090 0.82 CYP1B1 (0.46) ALDH1A1CES1MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed