SCHEMBL7361832

SCHEMBL7361832

CCOC(=O)c1c(C)cc(C)nc1CC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.50
CYP3A4 P08684 3/20 0.50
TDP1 Q9NUW8 1/20 0.50
ADORA3 P0DMS8 4/20 0.49
ALDH1A1 P00352 5/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 3/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46
MAPK1 P28482 1/20 0.46
KDM4E B2RXH2 4/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
GLA P06280 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
ATM Q13315 1/20 0.46
HSD17B10 Q99714 1/20 0.46
USP2 O75604 1/20 0.44
CA12 O43570 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24773784 0.87 SMN1; SMN2 (0.51) SMN1; SMN2CYP3A4TDP1ADORA3ALDH1A1
SCHEMBL7363101 0.87 ADORA3 (0.49) SMN1; SMN2CYP3A4TDP1ADORA3ALDH1A1
SCHEMBL7358402 0.85 CYP3A4 (0.49) SMN1; SMN2CYP3A4TDP1ADORA3ALDH1A1
SCHEMBL7362801 0.83 POLB (0.60) SMN1; SMN2CYP3A4TDP1ADORA3ALDH1A1
SCHEMBL10736055 0.81 SMN1; SMN2 (0.61) SMN1; SMN2CYP3A4TDP1ALDH1A1POLB
SCHEMBL25882373 0.81 ALDH1A1 (0.65) SMN1; SMN2CYP3A4ADORA3ALDH1A1POLB
SCHEMBL25878362 0.80 CYP3A4 (0.44) SMN1; SMN2CYP3A4TDP1ADORA3ALDH1A1
SCHEMBL11439946 0.80 SMN1; SMN2 (0.50) SMN1; SMN2CYP3A4TDP1ALDH1A1POLB
SCHEMBL11808110 0.80 KDM4E (0.52) SMN1; SMN2CYP3A4TDP1ALDH1A1POLB
SCHEMBL31644242 0.78 SMN1; SMN2 (0.52) SMN1; SMN2CYP3A4TDP1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805681-A4 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-05-06 EP disclosed
EP-0805681-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1997-11-12 EP disclosed
WO-1996022775-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-08-01 WO disclosed