SCHEMBL7361886

SCHEMBL7361886

CCOC=CC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
MAOB P27338 4/20 0.57
CES2 O00748 1/20 0.51
POLB P06746 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
P4HB P07237 1/20 0.45
SRD5A2 P31213 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
ADORA1 P30542 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24951715 0.82 ALDH1A1 (0.59) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL28630576 0.82 ALDH1A1 (0.59) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL10942203 0.82 ALDH1A1 (0.62) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL10942199 0.82 ALDH1A1 (0.62) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL9586253 0.79 ALDH1A1 (0.70) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL11461960 0.77 MAOB (0.68) ALDH1A1MAOBCES2POLBNPSR1
SCHEMBL10275631 0.77 AKT1 (0.54) ALDH1A1MAOBNPSR1MEN1KMT2A
SCHEMBL10439177 0.77 AKT1 (0.54) ALDH1A1MAOBNPSR1MEN1KMT2A
SCHEMBL10275628 0.77 AKT1 (0.54) ALDH1A1MAOBNPSR1MEN1KMT2A
SCHEMBL30786693 0.76 CES2 (0.61) ALDH1A1CES2POLBNPSR1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed